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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Rivista
Codice:
E022401
ISSN:
0960-894X
Dati Generali
Dati Generali
Pubblicazioni (135)
Pulisci
Ordina Pubblicazioni:
ascendente
decrescente
'Proximity frequencies' a new parameter to evaluate the profile of GABA
A
R modulators
Articolo
(-)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels
Articolo
1,2-Disubstituted Cyclohexane Derived Tripeptide Aldehydes as Novel Selective Thrombin Inhibitors
Articolo
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators.
Articolo
4-Connected azabicyclo[5.3.0]decane Smac mimetics-Zn2+ chelators as dual action antitumoral agents
Articolo
5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity.
Articolo
A New Lipophilic Fluorescent Probe for Interaction Studies of Bioactive Lipopeptides with Membrane Models
Articolo
A highly catalytically active ?-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules.
Articolo
A highly catalytically active gamma-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules
Articolo
A new cytotoxic tambjamine alkaloid from the Azorean nudibranch Tambja ceutae.
Articolo
A novel super-potent neurokinin a receptor antagonist containing dehydroalanine
Articolo
A novel thermophilic glycosynthase that effects branching glycosylation.
Articolo
An improved procedure for the synthesis of branched polyethylene glycols (pegs) with the reporter dipeptide Met-bala for protein conjugation
Articolo
Anchimeric assistance effect on regloselective hydrolysis of branched PEGs: a mechanistic investigation
Articolo
Anion inhibition studies of a beta-carbonic anhydrase from Clostridium perfringens
Articolo
Anion inhibition studies of the ?-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae.
Articolo
Anion inhibition studies of the beta-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae
Articolo
Anion inhibition studies of two new beta-carbonic anhydrases from the bacterial pathogen Legionella pneumophila
Articolo
Anion inhibition study of the beta-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis
Articolo
Arylboronic acids as dual-action FAAH and TRPV1 ligands
Articolo
Backbone modified formyl-methionyl tripeptide chemoattractants
Articolo
Beta-Casomorphins: Substitution of Phenylalanine with beta-homo Phenylalanine Increases the mu-Type Opioid Receptor Affinity
Articolo
Bradykinin antagonists modified with dipeptide mimetic beta-turn inducers
Articolo
Burkholderia pseudomallei gamma-carbonic anhydrase is strongly activated by amino acids and amines
Articolo
CARBONIC ANHYDRASE INHIBITORS: X-RAY CRYSTALLOGRAPHIC STUDIES FOR THE BINDING OF 5-AMINO-1,3,4-THIADIZOLE-2-SULFONAMIDE AND 5-(4-AMINO-3-CHLORO-5-FLUOROPHENYLSULFONAMIDO)-1,3,4-THIADIAZOLE-2-SULFONAMIDE TO HUMAN ISOFORM II
Articolo
Carbonic anhydrase VII is S-glutathionylated without loss of catalytic activity and affinity for sulfonamide inhibitors
Articolo
Carbonic anhydrase activators: Activation of the beta-carbonic anhydrase from Malassezia globosa with amines and amino acids
Articolo
Carbonic anhydrase inhibitors. Benzenesulfonamides incorporating cyanoacrylamide moieties strongly inhibit Saccharomyces cerevisiae beta-carbonic anhydrase
Articolo
Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.
Articolo
Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides - Solution and crystallographic studies
Articolo
Carbonic anhydrase inhibitors: Inhibition of the beta-class enzyme from the pathogenic yeast Candida glabrata with sulfonamides, sulfamates and sulfamides
Articolo
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II "selective" inhibitor celecoxib.
Articolo
Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II
Articolo
Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties
Articolo
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV.
Articolo
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of Thr200 and Gln92 for obtaining tight-binding inhibitors.
Articolo
Cloning, expression, purification and sulfonamide inhibition profile of the complete domain of the eta-carbonic anhydrase from Plasmodium falciparum
Articolo
Comparison of the sulfonamide inhibition profiles of the alpha-, beta- and gamma-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae
Articolo
Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide.
Articolo
Design of novel alpha7-subtype-preferring nicotinic acetylcholine receptor agonists: application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies
Articolo
Design, synthesis and biological evaluation of novel aminopropylcarboxamide derivatives as sigma ligands
Articolo
Design, synthesis and preliminary evaluation of
18
F-labelled 1,8-naphthyridin- and quinolin-2-one-3-carboxamide derivatives for PET imaging of CB2 cannabinoid receptor
Articolo
Development of mitochondrial-targeted derivatives o resveratrol.
Articolo
Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents.
Articolo
Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum-The eta-carbonic anhydrases
Articolo
Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands
Articolo
Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains.
Articolo
Discovery of potent nucleotide-mimicking competitive inhibitors of hepatitis C virus NS3 helicase.
Articolo
Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: towards the next generation HIV-1 inhibitors
Articolo
Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candidaalbicans and Candida glabrata
Articolo
Dual action Smac mimetics-zinc chelators as pro-apoptotic antitumoral agents
Articolo
Effect of acyclic monoterpene alcohols and their derivatives on TRP channels
Articolo
Efficient and chemoselective N-acylation of 10-amino-7-ethyl camptothecin with poly(ethylene glycol)
Articolo
Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants.
Articolo
Enantioselective synthesis and vanilloid activity evaluation of 1-beta-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks.
Articolo
Enantioselective synthesis and vanilloid activity evaluation of 1-â-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks
Articolo
Enzymatic regio- and diastereoselective hydrolysis of peracetylated glycerol- and erhythritol-beta-glucosides
Articolo
Enzymatic syntheses and selective hydrolysis of O-b-D-galactopyranosides using a marine mollusc b-galactosidase
Articolo
Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes.
Articolo
Evidences for complex formation between L-dabPNA and aegPNA
Articolo
Evidences for complex formation between l-dabPNA and aegPNA
Articolo
Expanding the chemical space of human serine racemase inhibitors
Articolo
Ganglioside GM1 mimics: Lipophilic substituents improve affinity for cholera toxin
Articolo
Glycosynthase-catalysed syntheses at pH below neutrality.
Articolo
Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors.
Articolo
Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB1 receptors
Articolo
Identification and in vitro characterization of a new series of potent and highly selective G9a inhibitors as novel anti-fibroadipogenic agents
Articolo
Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells.
Articolo
Impurity analysis of retinoic acid samples
Articolo
Indolyl-pyrrolone as a new scaffold for Pim1 inhibitors
Articolo
Indolyl-pyrrolone as a new scaffold for Pim1 inhibitors.
Articolo
Induction of erythroid differentation of human K562 cells by 3-O-acyl-1,2-O-isopropylidene-D-glucofuranose derivatives
Articolo
Inhibition of the R1 fragment of the cadmium-containing zeta-class carbonic anhydrase from the diatom Thalassiosira weissflogii with anions.
Articolo
Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates
Articolo
Kinetic and anion inhibition studies of a beta-carbonic anhydrase (FbiCA 1) from the C-4 plant Flaveria bidentis
Articolo
Marine bis-gamma-pyrone polypropionates of onchidione family and their effects on the XBP1 gene expression
Articolo
Metabolically labile cannabinoid esters: A 'soft drug' approach for the development of cannabinoid-based therapeutic drugs
Articolo
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds
Articolo
Molecular insights to the bioactive form of BV02, a reference inhibitor of 14-3-3? protein-protein interactions
Articolo
N-(thiazol-2-yl)-2-thiophene carboxamide derivatives as Abl inhibitors identified by a pharmacophore-based database screening of commercially available compounds.
Articolo
N-Hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: mode of binding in a complex with MMP-8.
Articolo
Natural and synthetic G-quadruplex interactive berberine derivatives.
Articolo
New aspartame-like sweeteners containing L-(alphaMe)Phe
Articolo
New highly hydrosoluble and not self-aggregated perylene derivatives with three and four polar side chains as G-quadruplex telomere targeting agents and telomerase inhibitors
Articolo
New metabolically stable fatty acid amide ligands of cannabinoid receptors: synthesis and receptor affinity studies
Articolo
New tetrazole-based selective anandamide uptake inhibitors.
Articolo
Novel imidazole-based combretastatin A-4 analogues: Evaluation of their in vitro antitumor activity and molecular modeling study of their binding to the colchicine site of tubulin
Articolo
One drug for two targets: Biological evaluation of antiretroviral agents endowed with antiproliferative activity
Articolo
Perylene diimides with different side chains are selective in inducing different G-Quadruplex DNA structures and in inhibiting telomerase
Articolo
Praziquantel derivatives I: Modification of the aromatic ring.
Articolo
Pyrazolo[3,4-d]pyrimidines-loaded human serum albumin (HSA) nanoparticles: Preparation, characterization and cytotoxicity evaluation against neuroblastoma cell line
Articolo
Rational design, synthesis and characterization of potent, drug-like monomeric Smac mimetics as pro-apoptotic anticancer agents
Articolo
Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition
Articolo
SYNTHESIS OF CARBAPENEMS VIA METALLOIMINES-ESTER ENOLATES CONDENSATION - A NEW SYNTHESIS OF (+)-1-BETA-METHYL PS-5
Articolo
Selective interactions of perylenederivatives having different side chains with inter- and intramolecular G-quadruplex DNA structures. A correlation with telomerase inhibition
Articolo
Soluble polyphenols: synthesis and bioavailability of 3,4',5-tri(alpha-D-glucose-3-O-succinyl)resveratrol.
Articolo
Structure-activity relationships of the prototypical TRPM8 agonist icilin
Articolo
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The homovanillyl moiety
Articolo
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene
Articolo
Sulfonamide inhibition profile of the gamma-carbonic anhydrase identified in the genome of the pathogenic bacterium Burkholderia pseudomallei the etiological agent responsible of melioidosis
Articolo
Sulfonamide inhibition studies of the delta-carbonic anhydrase from the diatom Thalassiosira weissflogii
Articolo
Sulfonamide inhibition studies of the gamma-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea
Articolo
Sulfonamide inhibition studies of the gamma-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis
Articolo
Sulfonamide inhibition studies of the gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis
Articolo
Sulfonamide inhibition study of the beta-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans
Articolo
Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers.
Articolo
Synthesis and alpha4beta2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes.
Articolo
Synthesis and anticonvulsant activity of new N-1',N-3'-disubstituted-2'H,3H,5'H-spiro-(2-benzofuran-1,4'-imidazolidine)-2',3,5'-triones
Articolo
Synthesis and binding affinity at alpha4beta2 and alpha7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system
Articolo
Synthesis and biological characterization of 3-(imidazol-1-ylmethyl)piperidine sulfonamides as aromatase inhibitors
Articolo
Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators
Articolo
Synthesis and biological evaluation of cyclic and branched peptide analogues as ligands for cholecystokinin type 1 receptor
Articolo
Synthesis and biological evaluation of new potential inhibitors of N-acylethanolamine hydrolyzing acid amidase.
Articolo
Synthesis and biological evaluation of novel amides of dopamine with polyunsaturated fatty acids
Articolo
Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands
Articolo
Synthesis and biological investigation of S-aryl-S-DABO derivatives as HIV-1 inhibitors.
Articolo
Synthesis and enzymatic evaluation of novel partially fluorinated thiol dual ACE/NEP inhibitors
Articolo
Synthesis and evaluation of diverse thio avarol analogs as potential UVB photoprotective candidates
Articolo
Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors
Articolo
Synthesis and preliminary biological profile of new NO-donor tolbutamide analogues
Articolo
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors
Articolo
Synthesis of All-trans Isomer of Arachidonic Acid and Its Effect on Rabbit Plateled Aggregation
Articolo
Synthesis of a potential photoactivatable anandamide analog
Articolo
Synthesis of hybrid distamycin-cysteine labeled with Tc-99m: a model for a novel class of cancer imaging agents
Articolo
Synthesis of new Praziquantel analogues: Potential candidates for the treatment of schistosomiasis
Articolo
Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis gamma-carbonic anhydrase
Articolo
Synthetic approaches to DNMT inhibitor SGI-1027 and effects on the U937 leukemia cell line.
Articolo
TRPA1 channels as targets for resveratrol and related stilbenoids
Articolo
Tetrahydro-beta-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels. .
Articolo
The extremo-?-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines
Articolo
The zinc coordination pattern in the eta-carbonic anhydrase from Plasmodium falciparum is different from all other carbonic anhydrase genetic families
Articolo
Towards novel S-DABOC inhibitors: Synthesis, biological investigation, and molecular modeling studies.
Articolo
Trehalose-based neuroprotective autophagy inducers
Articolo
Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore
Articolo
omega-Alkoxy analogues of SAHA(vorinostat) as inhibitors of HDAC: a study of chain-lenght and stereochemical dependence.
Articolo
No Results Found
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