Enanthioselective synthesis of protected D-serine from tetrahydrooxazin-4-one via hetero Diels-Alder reaction
Articolo
Data di Pubblicazione:
2002
Abstract:
Hetero Diels-Alder reaction between 2-aza-3-trimethylsilyloxy-1,3-diene and aldehydes gives rise to tetrahydrooxazin-4-ones, useful intermediates in the synthesis of alpha-amino-beta-hydroxy acids. Herein we report the complete stereoselective synthesis of D-serine Cbz-methyl ester.
Tipologia CRIS:
01.01 Articolo in rivista
Keywords:
ALPHA-AMINO-ACIDS; PRACTICAL STEREOSELECTIVE SYNTHESIS; BETA-HYDROXY; DIASTEREOSELECTIVE SYNTHESIS; ELECTROPHILIC AMINATION; ASYMMETRIC-SYNTHESIS; DERIVATIVES; THREONINES; RECEPTOR; ESTERS
Elenco autori:
Panunzio, Mauro; Bandini, Elisa
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